78322 2,3-Oxidosqualene-lanosterol cyclase inhibitor 125857 3 Hydroxyanthranilate oxygenase inhibitor 25482 5 Alpha reductase inhibitor 8283 5 Hydroxytryptamine 1 agonist 14271 5 Hydroxytryptamine 1 antagonist 10341 5 Hydroxytryptamine 1A agonist 13523 5 Hydroxytryptamine 1A antagonist 22575 5 Hydroxytryptamine 1B agonist 7933 5 Hydroxytryptamine 1D agonist 24908 5 Hydroxytryptamine 1D antagonist 12084 5 Hydroxytryptamine 1F agonist 110948 5 Hydroxytryptamine 2 agonist 16366 5 Hydroxytryptamine 2 antagonist 18564 5 Hydroxytryptamine 2A antagonist 55821 5 Hydroxytryptamine 2B antagonist 123651 5 Hydroxytryptamine 2C agonist 32114 5 Hydroxytryptamine 2C antagonist 91279 5 Hydroxytryptamine 3 agonist 8728 5 Hydroxytryptamine 3 antagonist 8854 5 Hydroxytryptamine 4 agonist 13442 5 Hydroxytryptamine 4 antagonist 10285 5 Hydroxytryptamine agonist 20447 5 Hydroxytryptamine antagonist 116635 5 Hydroxytryptamine release stimulant 17651 5 Hydroxytryptamine uptake inhibitor 119501 ADP ribosyl transferase inhibitor 60581 AMPA receptor agonist 28646 AMPA receptor antagonist 34136 Acetyl CoA transferase inhibitor 35115 Acetylcholine M1 receptor agonist 59781 Acetylcholine M2 receptor antagonist 63401 Acetylcholine M3 receptor antagonist 54873 Acetylcholine agonist 50602 Acetylcholine antagonist 45884 Acetylcholine muscarinic agonist 49179 Acetylcholine muscarinic antagonist 16738 Acetylcholine neuromuscular blocking agent 78391 Acetylcholine nicotinic agonist 57340 Acetylcholine nicotinic antagonist 118820 Acetylcholine release stimulant 46026 Acetylcholinesterase inhibitor 66813 Acute neurologic disorders treatment 13151 Adenosine A1 receptor agonist 25406 Adenosine A1 receptor antagonist 8460 Adenosine A2 receptor agonist 16326 Adenosine A2 receptor antagonist 35017 Adenosine A2a receptor agonist 24353 Adenosine A2a receptor antagonist 9116 Adenosine A3 receptor agonist 130827 Adenosine A3 receptor antagonist 13123 Adenosine deaminase inhibitor 50463 Adenosine kinase inhibitor 8501 Adenosine receptor agonist 21556 Adenosine receptor antagonist 40787 Adrenaline agonist 23473 Adrenaline antagonist 90977 Adrenergic transmitter uptake inhibitor 123685 Alcohol dehydrogenase inhibitor 41737 Aldose reductase inhibitor 90205 Aldosterone antagonist 54036 Alkylator 39936 Alkylphospholipid 108376 Alpha 1 adrenoreceptor agonist 14503 Alpha 1 adrenoreceptor antagonist 72576 Alpha 2 adrenoreceptor agonist 22644 Alpha 2 adrenoreceptor antagonist 50524 Alpha adrenoreceptor agonist 21666 Alpha adrenoreceptor antagonist 26458 Alpha glucosidase inhibitor 125412 Alzheimer's disease treatment 117119 Aminopeptidase microsomal inhibitor 72827 Anabolic 88415 Analeptic 50193 Analgesic 53160 Analgesic, non-opioid 20281 Analgesic, opioid 45435 Anaphylatoxin receptor antagonist 37004 Androgen agonist 41125 Androgen antagonist 64811 Anesthetic 90448 Anesthetic general 98892 Anesthetic inhalation 63042 Anesthetic local 89266 Angiogenesis inhibitor 2874 Angiotensin AT1 receptor antagonist 19067 Angiotensin AT2 receptor antagonist 7831 Angiotensin II receptor antagonist 7831 Angiotensin antagonist 9392 Angiotensin converting enzyme inhibitor 83807 Anorexic 66284 Anti-Helicobacter pylori 39225 Antiacne 53209 Antiallergic 116395 Antiamebic 60526 Antianginal 41061 Antiarrhythmic 70669 Antiarthritic 113212 Antiasthmatic 53378 Antibacterial 12512 Antibiotic 16115 Antibiotic Aminoglycoside-like 5389 Antibiotic Anthracycline-like 4544 Antibiotic Carbacephem-like 1699 Antibiotic Carbapenem-like 1378 Antibiotic Cephalosporin-like 2557 Antibiotic Glycopeptide-like 2931 Antibiotic Isocephem-like 3237 Antibiotic Macrolide-like 2446 Antibiotic Naphthyridine-like 16116 Antibiotic Oxacephem-like 5395 Antibiotic Oxazolidinone-like 1166 Antibiotic Penem-like 1793 Antibiotic Penicillin-like 818 Antibiotic Quinolone-like 3469 Antibiotic Rifamycin-like 11736 Antibiotic Tetracycline-like 6550 Antibiotic Tribactam-like 16907 Antibiotic Trimethoprim-like 3401 Antibiotic beta Lactam-like 93881 Anticataract 63327 Anticerebroischemic 9216 Anticholelithogenic 22848 Anticoagulant 89902 Anticoccidial 73899 Anticonvulsant 31683 Antidepressant 56910 Antidepressant, Imipramin-like 50210 Antidiabetic 69584 Antidiabetic symptomatic 11646 Antidiuretic hormone antagonist 118192 Antidyskinetic 16914 Antiemetic 30343 Antiemphysemic 81997 Antifungal 56989 Antiglaucomic 101633 Antihelmintic 13139 Antihistaminic 94584 Antihypercholesterolemic 54533 Antihypertensive 101282 Antiinfective (HIV) 22788 Antiinfertility, female 91004 Antiinflammatory 9078 Antiinflammatory steroid 120912 Antiinflammatory, intestinal 101384 Antiinflammatory, pancreatic 109787 Antiischemic 128333 Antilipidemic 73790 Antimalarial 38376 Antimetabolite 18285 Antimigraine 31592 Antimitotic 4533 Antimitotic Taxane-like 8381 Antimitotic podophyllotoxin-like 101193 Antimycobacterial 38236 Antimycoplasmal 93344 Antineoplastic 29103 Antineoplastic alkaloid 33233 Antineoplastic antibiotic 52923 Antineoplastic enhancer 38600 Antiobesity 48035 Antiosteoporotic 65603 Antioxidant 54447 Antiparkinsonian 104439 Antiparkinsonian, rigidity relieving 84044 Antiparkinsonian, tremor relieving 82402 Antiprotozoal 123771 Antipruritic 83547 Antipsoriatic 19677 Antipsychotic 128643 Antiseptic 107061 Antismoking 74248 Antispirochetal 105438 Antitoxic 111742 Antitrichomonal 106559 Antitrypanosomal 68966 Antitussive 61262 Antitussive, narcotic 76261 Antiulcerative 74185 Antiviral 43885 Antiviral (HIV) 124605 Antiviral (hepatitis C) 136815 Antiviral (hepatitis) 6285 Antiviral (influenza) 33921 Anxiolytic 17736 Aromatase inhibitor 125520 Arrhythmogenic 115560 Atherosclerosis treatment 16492 Atrial natriuretic polypeptide agonist 23320 Benzodiazepine agonist 55923 Benzodiazepine agonist partial 79764 Benzodiazepine antagonist 39436 Benzodiazepine inverse agonist 36024 Beta 1 adrenoreceptor agonist 19933 Beta 1 adrenoreceptor antagonist 23920 Beta 2 adrenoreceptor agonist 5942 Beta 3 adrenoreceptor agonist 23679 Beta adrenoreceptor agonist 25085 Beta adrenoreceptor antagonist 26732 Beta lactamase inhibitor 11814 Bisphosphonate 6259 Bombesin antagonist 93757 Bone formation stimulant 75675 Bone resorption inhibitor 10305 Bradykinin B2 receptor antagonist 12330 Bradykinin antagonist 40654 Bronchodilator 92495 CNS active muscle relaxant 22956 Calcium agonist 44273 Calcium channel antagonist 91887 Calcium regulator 88529 Calmodulin antagonist 77045 Calpain inhibitor 108009 Cannabinoid receptor agonist 6454 Carbonic anhydrase inhibitor 111451 Carcinogenic 85284 Cardiodepressant 116011 Cardioprotectant 46305 Cardiotonic 124907 Cardiotoxic 118955 Cardiovascular analeptic 119575 Catechol O methyltransferase inhibitor 36821 Cathepsin B inhibitor 119478 Cathepsin L inhibitor 131871 Chemopreventive 52688 Chemoprotective 39499 Cholecystokinin A agonist 21548 Cholecystokinin A antagonist 23234 Cholecystokinin B antagonist 12858 Cholecystokinin agonist 15471 Cholecystokinin antagonist 87711 Choleretic 71648 Cholesterol esterase inhibitor 107629 Cholinergic agonist 44475 Cholinergic antagonist 2721 Chymotrypsin inhibitor 90793 Coagulant 110505 Cocain dependency treatment 51364 Cognition disorders treatment 17431 Collagenase inhibitor 106648 Complement inhibitor 73033 Contraceptive 82027 Corneal wound healing stimulator 6395 Corticosteroid-like 38040 Cyclooxygenase 2 inhibitor 77575 Cyclooxygenase inhibitor 107204 Cystic fibrosis treatment 121334 Cytokine modulator 109328 Cytosole dipeptidase inhibitor 113439 Cytostatic 36092 DNA intercalator 78100 Dermatologic 18282 Dihydrofolate reductase inhibitor 98436 Dihydroorotate dehydrogenase inhibitor 71067 Dipeptidyl aminopeptidase IV inhibitor 72449 Diuretic 114490 Dopa decarboxylase inhibitor 9290 Dopamine D1 agonist 20577 Dopamine D1 antagonist 8312 Dopamine D2 agonist 12266 Dopamine D2 antagonist 12715 Dopamine D3 antagonist 9954 Dopamine D4 antagonist 21487 Dopamine agonist 11970 Dopamine antagonist 7942 Dopamine autoreceptor agonist 40178 Dopamine beta hydroxylase inhibitor 44719 Dopamine uptake inhibitor 29079 Elastase inhibitor 119411 Embryotoxic 26196 Endothelin A receptor antagonist 16976 Endothelin B receptor antagonist 110482 Endothelin antagonist 20008 Endothelin receptor antagonist 25794 Endothelin-converting enzyme inhibitor 14037 Enkephalinase inhibitor 136247 Erythropoietin 22553 Estrogen agonist 29153 Estrogen antagonist 13648 Estrogen receptor modulator 66903 Estrone sulfatase inhibitor 89867 Excitatory amino acid agonist 96878 Excitatory amino acid antagonist 89481 Expectorant 55950 Factor VIIa inhibitor 42552 Factor XIIIa inhibitor 8377 Factor Xa inhibitor 27572 Farnesyltransferase inhibitor 81942 GABA A receptor agonist 77515 GABA A receptor antagonist 98060 GABA B receptor agonist 64771 GABA B receptor antagonist 75751 GABA aminotransferase inhibitor 98491 GABA receptor agonist 86697 GABA receptor antagonist 49393 GABA uptake inhibitor 6769 GP IIb/IIIa receptor antagonist 54400 Gastric antisecretory 15916 Gastrin inhibitor 5369 Gastrin-releasing peptide antagonist 119193 Geranylgeranyltransferase inhibitor 96539 Glucagon receptor antagonist 7592 Glucocorticoid agonist 34362 Glucocorticoid antagonist 78872 Glucose-6-phosphate translocase inhibitor 26360 Glutamate (mGluR) agonist 76230 Glutamate (mGluR) antagonist 50033 Glutamate (mGluR1) agonist 44436 Glutamate (mGluR1) antagonist 68962 Glutamate (mGluR1a) agonist 74939 Glutamate (mGluR2) agonist 61888 Glutamate (mGluR2) antagonist 64840 Glutamate (mGluR3) agonist 75397 Glutamate (mGluR3) antagonist 86960 Glutamate (mGluR5) agonist 122055 Glutamate (mGluR5) antagonist 68962 Glutamate (mGluR5a) agonist 37730 Glutamate (mGluR6) agonist 80042 Glutamate (mGluR6) antagonist 37312 Glutamate receptor agonist 44820 Glutamate receptor antagonist 73583 Glutamate uptake inhibitor 9691 Glycinamide ribonucleotide formyltransferase inhibitor 105554 Glycine receptor agonist 6339 Growth hormone release promoting 18254 Growth hormone secretion inhibitor 60372 Growth stimulant 72332 Gynecological disorders treatment 45448 H+/K+-transporting ATPase inhibitor 125865 HCV NS3 protease inhibitor 29411 HCV NS3-4A protease inhibitor 86908 HCV NS3-helicase inhibitor 90545 HCV serine protease inhibitor 99253 HDL-cholesterol increasing 128170 HIV integrase inhibitor 20743 HIV protease inhibitor 11976 HIV-1 protease inhibitor 12864 HMG CoA reductase inhibitor 48197 HMG CoA synthase inhibitor 64675 Hair growth promoter 51945 Hematopoietic 124606 Hematopoietic inhibitor 79423 Hepatoprotectant 121204 Hestagen antagonist 9438 Hestagen-like 74136 Histamine H1 receptor antagonist 88845 Histamine H2 receptor agonist 26317 Histamine H2 receptor antagonist 39657 Histamine H3 receptor agonist 4322 Histamine H3 receptor antagonist 37062 Histamine agonist 31867 Histamine antagonist 122281 Histamine release stimulant 58982 Histidine decarboxylase inhibitor 79971 Hypertensive 104416 Hypertensive, ophthalmic 96751 Hypertermic 136486 Hypnotic 74042 Hypoglycemic 52079 Hypolipemic 94912 Hypotermic 63437 Ileal bile acid transport inhibitor 77450 Immunomodulator 72345 Immunostimulant 80505 Immunosuppressant 4714 Immunosuppressant Cyclosporine-like 66201 Inflammatory Bowel disease threatment 101398 Insulin promoter 68412 Insulin secretagoues 91980 Interferon inducer 102163 Interleukin 1 antagonist 16380 Interleukin 1 beta converting enzyme inhibitor 138169 Interleukin 6 antagonist 71753 Interleukin 8 antagonist 16380 Interleukin agonist 99908 Interleukin antagonist 52373 Irritable Bowel syndrome therapy 59070 Kainate receptor agonist 63449 Kainate receptor antagonist 139738 Keratolytic 132927 Keratoses actinic(solar) treatment 138938 Leukopoiesis inhibitor 17700 Leukotriene A4 hydrolase inhibitor 24340 Leukotriene B4 antagonist 13790 Leukotriene D4 antagonist 33605 Leukotriene antagonist 43792 Leukotriene synthesis inhibitor 68821 Lipid peroxidase inhibitor 44136 Lipoxygenase inhibitor 95452 Liver fibrosis treatment 6957 Luteinizing hormone-releasing hormone agonist 7901 Luteinizing hormone-releasing hormone antagonist 83569 Lymphocytopoiesis inhibitor 82221 MAO inhibitor 70015 MAO-A inhibitor 44380 MAO-B inhibitor 91623 Maillard reaction inhibitor 111291 Male reproductive disfunction treatment 89433 Mannosidase inhibitor 21851 Matrix metalloproteinase inhibitor 79415 Mediator release inhibitor 24233 Melatonin agonist 123047 Melatonin antagonist 135805 Metabolic 45805 Microtubule formation inhibitor 16171 Mineralocorticoid 100634 Miotic 11764 Motilin-like 77975 Mucolytic 101496 Multiple sclerosis treatment 80050 Muscle relaxant 104089 Mutagenic 39413 Mydriatic 104636 Myocardial ischemia treatment 7553 Myristoyl transferase inhibitor 70305 NMDA receptor agonist 40521 NMDA receptor antagonist 116190 NMDA receptor glycine site agonist 56719 NMDA receptor glycine site antagonist 93920 NMDA receptor polyamine site activator 28544 NMDA receptor polyamine site blocker 70660 Narcotic antagonist 103174 Nasal decongestant 16732 Neuraminidase (influenza) inhibitor 10580 Neurokinin 2 antagonist 13467 Neurokinin 3 antagonist 6411 Neurokinin antagonist 47487 Neuropeptide Y antagonist 47487 Neuropeptide antagonist 31194 Neurotensin receptor antagonist 103957 Neurotrophic factor 6654 Neutral endopeptidase inhibitor 27648 Nitric oxide donor 57706 Nitric oxide synthase inhibitor 118762 Non-steroidal antiinflammatory agent 113354 Nootropic 119931 Nucleotide metabolism regulator 38584 O6-alkylguanine-DNA alkyltransferase inhibitor 67044 Ophthalmic drug 10308 Opioid agonist 46033 Opioid antagonist 12121 Opioid delta receptor agonist 12729 Opioid kappa receptor agonist 31484 Opioid mu receptor agonist 52696 Opioid partial agonist 68204 Ornithine decarboxylase inhibitor 66957 Oxytocin agonist 48416 Oxytocin antagonist 48908 Pancreatic disorders treatment 95400 Parathyroid hormone antagonist 24833 Peristaltic stimulant 67825 Phosphodiesterase I inhibitor 41008 Phosphodiesterase III inhibitor 26075 Phosphodiesterase IV inhibitor 57422 Phosphodiesterase V Inhibitor 26978 Phosphodiesterase inhibitor 54489 Phospholipase A2 inhibitor 126345 Phospholipase C inhibitor 55574 Phospholipase inhibitor 58616 Photosensitizer 24271 Platelet activating factor antagonist 124440 Platelet adhesion inhibitor 39626 Platelet aggregation inhibitor 110045 Platelet antagonist 125977 Poly(ADP-ribose)synthethase inhibitor 58036 Postcoital contraceptive 22054 Potassium channel activator 58182 Potassium channel antagonist 12972 Progesterone antagonist 63373 Progestin agonist 86409 Prolactin inhibitor 24306 Prolactin secretion inhibitor 14197 Prolyl endopeptidase inhibitor 32059 Prostaglandin E2 antagonist 10889 Prostaglandin agonist 87999 Prostaglandin antagonist 37602 Prostate disorders treatment 30851 Protease inhibitor 59070 Protein kinase C inhibitor 42833 Protocollagen prolyl hydroxylase inhibitor 100680 Psychosexual dysfunction treatment 91057 Psychostimulant 40843 Psychotropic 14395 Purine nucleoside phosphorylase inhibitor 3110 Purinergic P2 agonist 39588 Purinergic P2 antagonist 22392 Purinergic P2T antagonist 3110 Purinergic receptor agonist 39588 Purinergic receptor antagonist 80660 Quisqualate antagonist 102815 Radioprotector 106870 Radiosensitizer 19058 Reductant 57291 Renal disease treatment 3291 Renin inhibitor 90351 Respiratory analeptic 94021 Respiratory distress syndrome treatment 56144 Restenosis treatment 11136 Retinoid-like 60924 Reverse transcriptase inhibitor 69596 Rhinitis treatment 26428 Ribonucleoside diphosphate reductase inhibitor 51050 Ribonucleotide reductase inhibitor 11925 S-adenosyl-L-homocysteine hydrolase inhibitor 121393 S-adenosyl-L-methionine decarboxylase inhibitor 81979 Saluretic 56705 Saluretic, reabsorbtion inhibitor 114830 Sclerosant 82786 Sedative 20438 Selectin antagonist 72087 Septic shock treatment 21221 Sigma receptor antagonist 39678 Signal transduction pathways inhibitor 81573 Skeletal muscle relaxant 96734 Sodium channel blocker 118432 Sodium channel blocker class Ib 4228 Somatostatin agonist 66792 Spasmogenic 62854 Spasmolytic 73354 Spasmolytic, Papaverin-like 75092 Spasmolytic, urinary 139227 Spermicide 68408 Squalene epoxidase inhibitor 21851 Squalene synthetase inhibitor 6672 Steroid-like 9415 Substance P antagonist 78283 Succinic dehydrogenase inhibitor 41611 Sulfonylureas 92785 Sympatholytic 130176 TNF-alpha release inhibitor 121411 Teratogen 121411 Teratogen and/or embryotoxic 22959 Thiol protease inhibitor 8157 Thrombin inhibitor 98495 Thrombolytic 25638 Thromboxane antagonist 27512 Thromboxane synthase inhibitor 121706 Thymidine kinase inhibitor 17802 Thymidylate synthase inhibitor 55473 Thyroid hormone agonist 79822 Thyroid hormone antagonist 16993 Thyrotropin releasing hormone agonist 141786 Topoisomerase II inhibitor 41087 Topoisomerase inhibitor 45047 Treponemicidal 30236 Trypsin inhibitor 27755 Tryptase inhibitor 56928 Tumour necrosis factor antagonist 60942 Tyrosine kinase inhibitor 97957 Ulcerogenic 125594 Uricosuric 58348 Uridine phosphorylase inhibitor 53091 Urinary incontinence treatment 107518 Urokinase inhibitor 22762 Uterine relaxant 10331 Uterine stimulant 65667 Vasodilator 25318 Vasopressin 1 antagonist 9020 Vasopressin 2 antagonist 84040 Vasopressor 100146 Vitamin 3024 Vitamin D-like 116061 Xanthine oxidase inhibitor 7443 Xanthine-like 22543 cAMP modulator 102235 cAMP phosphodiesterase inhibitor